| ORGN | Thursday, August 23, 2007 | ||
8:00 AM-12:00 PM BCEC -- 254 A/B, Oral | |||
Heterocycles and Aromatics | |||
| Presiding: | Scott McN. Sieburth | ||
| 8:00 AM | 933 | A new and efficient preparation of 2-aminothiazole-5-carbamides, applications to the synthesis of Dasatinib, a new potent pan-src kinase inhibitor Bang-Chi Chen, Rulin Zhao, Bei Wang, Robert Droghini, Jean Lajeunesse, Pierre Sirard, Masaki Endo, Balu Balasubramanian, Joel C Barrish | |
| 8:20 AM | 934 | Kilogram synthesis of a LFA-1/ICAM inhibitor Albert J. DelMonte | |
| 8:40 AM | 935 | A regiospecific synthesis of N-aryl and N-alkyl benzimidazoles Nan Zheng, Kevin W. Anderson, Xiaohua Huang, Hanh Nho Nguyen, Stephen L. Buchwald | |
| 9:00 AM | 936 | Origins of selectivity in Pd-catalyzed C-N bond-forming reactions using biarylphosphine ligands Mark R. Biscoe, Timothy E. Barder, Stephen L. Buchwald | |
| 9:20 AM | 937 | Combined directed metalation and cross coupling tactics: A new carbanionic indole N-carbamoyl translocation reaction Victor Snieckus, Katherine A. Groom, Zhongdong Zhao | |
| 9:40 AM | 938 | Highly regioselective syntheses of N1-substituted and N2-substituted 1,2,3-triazoles Sen Wai Kwok, Jason Hein, Valery V. Fokin, K. Barry Sharpless | |
| 10:00 AM | 939 | Isomeric diazadienes via the Lewis acid-mediated isomerization of methylenecyclopropyl hydrazones Mark E. Scott, Yann Bethuel, Mark Lautens | |
| 10:20 AM | 940 | Tandem benzannulation cyclization strategy for the synthesis of highly-substituted indoles Tin Yiu Lam, Rick L. Danheiser | |
| 10:40 AM | 941 | Tandem benzannulation ring-closing metathesis strategy for the synthesis of benzo-fused nitrogen heterocycles Xiao Yin Mak, Aimee L. Crombie, Rick L. Danheiser | |
| 11:00 AM | 942 | What are the requirements for monohomoaromatic carbocations with ≥10 π electrons? A DFT study Philip M. Warner | |
| 11:20 AM | 943 | What is the π electron size limit for neutral bishomoaromaticity?: a DFT study Philip M. Warner | |
| 11:40 AM | 944 | N-Heterocyclic carbene (NHC) catalyzed synthesis of isoxazolidin-5-ones and a one-pot synthesis of β-amino acid esters Jayasree Seayad, Pranab K. Patra, Yugen Zhang, Jackie Y Ying | |
Heterocycles and Aromatics -- Next Session
Symposium Grid -- Division of Organic Chemistry -- Session Listing
The 234th ACS National Meeting, Boston, MA, August 19-23, 2007