Synthesis and biological activity of some C- and N- alkylated derivatives of 3-methyl quinoxaline-2-one

ORGN 785

Anita R Mali, orgchem_anitamali2004@yahoo.co.in and MB. Deshmukh, m_deshmukh1@rediffmail.com. department of chemistry, Shivaji University, kolhapur, Maharashtra, kolhapur, IN 416004, India
Abstract: Quinoxaline derivatives are very useful compounds with well-known biological activity. Whereas quinoxaline compounds are important components of several pharmacologicaly active moieties. Certain quinoxaline 2,3 diones and quinoxaline 2-ones were highly potent NMDA receptor antagonists. Also quinoxaline based materials were used as ETLs or (Electron transporting layer) or hole blocking layers in OLEDs (organic light emitting diodes). Hence, due to this commendable biological activity the synthesis of some new derivatives of 3-methyl-2-one quinoxalines was reported.

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