| MEDI | Wednesday, 13 September 2006 | ||
8:30 AM-12:30 PM Moscone Center -- Room 102, Oral | |||
Neuropeptide GPCRs | |||
| Sponsored by Teledyne Isco | |||
| Organizers: | Jeff Chen Robert DeVita Robert Ring | ||
| 8:30 AM | 302 | Design and development of vasopressin V1a antagonists Christophe D. Guillon, Michael Brownstein, Craig F. Ferris, Shi-Fang Lu, Karine Fabio, Marvin J. Miller, Ned D. Heindel, Neal G. Simon, Gary A. Koppel | |
| 9:10 AM | 303 | Novel diketopiperazines as potent and selective oxytocin antagonists John Liddle, Deirdre M B Hickey, Simon Peace, Alan D Borthwick, Patrick M Woollard, Michael J Allen, David P Brooks | |
| 9:50 AM | 304 | Development of Bradykinin B1 receptor antagonists as novel analgesics Scott D. Kuduk | |
| 10:30 AM | 305 | Discovery of novel Bradykinin B1 receptor antagonists for the treatment of pain and inflammation Wenyuan Qian, Kaustav Biswas, Toshihiro Aya, Joe Zhu, Tanya Peterkin, Jason Human, Jian Chen, Benny C. Askew, Leyla Arik, Eileen Johnson, Rich Loeloff, Ming Huang, Hong Dong, Barton Manning, Gondi Kumar, Smriti Joseph, Janan Jona | |
| 11:10 AM | 306 | Strategies and tactics for lead optimization of melanin concentrating hormone receptor 1 antagonists Philip R. Kym, Andrew J. Souers, John K. Lynch, Rajesh Iyengar, Andrew S. Judd, Anil Vasudevan, Ju Gao, Jennifer C. Freeman, Dariusz Wodka, Mathew Mulhern, Gang Zhao, James Polakowski, Thomas J. Campbell, Jason A. Segreti, Glenn A. Reinhart, Ryan M. Fryer, Lee Pruesser, Sevan Brodjian, Brian D. Dayton, Dennis G. Fry, Doug H. Falls, Regina M. Reilly, Kennan C. Marsh, Lisa E. Hernandez, Christoper Blackburn, Jennifer Lee Che, Courtney Cullis, Sujen Lai, Matthew J. Lamarche, Martin Maguire, Michael Brune, Eugene N. Bush, Robin Shapiro, Victoria Knourek-Segel, Hing L. Sham, Christine A. Collins | |
| 11:50 AM | 307 | The discovery of heterocyclic MCH R1 antagonists Donald L Hertzog, Kamal A Al-Barazanji, Kevin K Barvian, Eric C Bigham, Michael J Bishop, Christy S Britt, David L Carlton, Andrew J Carpenter, Joel P Cooper, Dulce M Garrido, Aaron S Goetz, Gary M Green, Mary K Grizzle, Yu C Guo, Anthony L Handlon, Clifton E Hyman, Diane M Ignar, Daniel G Lang, Ronda O Morgan, Andrew J Peat, Gregory E Peckham, Amy J Reisinger, Jason D Speake, Will R Swain, Francis X Tavares, Huiqiang Zhou | |
Symposium Grid -- Division of Medicinal Chemistry -- Session Listing
Symposium Grid -- Drug Discovery -- Session Listing
The 232nd ACS National Meeting, San Francisco, CA, September 10-14, 2006