ORGN 503 |
| A one-pot method for preparing the oxazolidinone acetamide 4 in excellent yield has been developed. This method employs the mesylate 1a rather than the comparatively more expensive nosylate 1b. The use of commercially available sodium diformylamide as the nitrogen source overcomes problematic secondary amine formation and the use of highly toxic and explosive reagents.
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New Reactions and Methodology, Heterocycles and Aromatics, Bioorganic Chemistry
8:00 PM-10:00 PM, Tuesday, 12 September 2006 Moscone Center -- Hall D, Poster
Division of Organic Chemistry |
