MEDIMonday, 27 March 2006

9:00 AM-12:35 PM Georgia World Congress Center -- Georgia Ballroom 3, Oral
Novel Antithrombotic Agents
Sponsored by Teledyne Isco
Organizer, Presidings:Christopher Bigge
Mimi L. Quan
9:00 AMIntroductory Remarks
9:05 AMLead generation and optimization strategies for the development of orally efficacious fXa inhibitors
Michael R. Wiley
Paper Withdrawn
10:15 AMDesign and synthesis of novel himbacine based thrombin receptor (Par-1) antagonists
Mariappan V. Chelliah, Samuel Chackalamannil, Yan Xia, Keith Eagen, Hsingan Tsai, Martin Clasby, Xiaobang Gao, William J. Greenlee, Ho-Sam Ahn, George Boykow, Carolyn Foster, Yunsheng Hsieh, Jacqueline Agans-Fantuzzi, Matthew Bryant, Madhu Chintala
10:50 AMDesign and synthesis of a novel orally efficacious PAI-1 inhibitor for the treatment of fibrinolytic impairment
Scott C. Mayer, Thomas Antrilli, Ann Aulabaugh, John A. Butera, David L. Crandall, Hassan Elokdah, Stephen Gardell, Eric Gundersen, James K. Hennan, Girija Krishnamurthy, Geraldine R. McFarlane, Gwen Morgan, Robert Swillo
11:25 AMTAFIa Inhibitors for treatment of thrombosis
Julian Blagg
12:00 PMConcluding Remarks

Symposium Grid -- Division of Medicinal Chemistry -- Session Listing

Symposium Grid -- Drug Discovery -- Session Listing

The 231st ACS National Meeting, Atlanta, GA, March 26-30, 2006