| MEDI | Sunday, 26 March 2006 | ||
1:30 PM-5:00 PM Georgia World Congress Center -- Georgia Ballroom 1, Oral | |||
First Time Disclosure of Clinical Candidates | |||
| Sponsored by Wyeth Research | |||
| Organizer: | Balu Balasubramanian | ||
| 1:30 PM | 17 | Discovery and development of a small molecule antagonist of leukocyte function-associated antigen-1 (LFA-1) Murali T. G. Dhar, Suzanne J. Suchard, Dominique Potin, Michèle Launay, Francoise Monatlik, Patrice Malabre, Maud Fabreguettes, André Fouquet, Magali Maillet, Eric Nicolaï, Loïc Dorgeret, François Chevallier, Dominique Besse, Monique Dufort, François Caussade, Dawn K. Stetsko, Stacey Skala, Patricia M. Davis, Praveen Balimane, Karishma Patel, Zheng Yang, Punit Marathe, Pathanjali Kadiyala, Kim W. Mcintyre, Xiaoxia Yang, Jennifer Postelneck, Robert Townsend, Sam Chao, Leslie Leith, Zili Xiao, Arvind Mathur, Bang-Chi Chen, Daugh-Rurng Wu, Ravindra Tejwani, Denette Murphy, Russell S. Weiner, Murray McKinnon, Stephen Bai, Joel C. Barrish, Jeffrey A. Robl, Edwin J. Iwanowicz | |
| 2:05 PM | 18 | Design and synthesis of potent, selective, and orally efficacious DPP4 inhibitors accelerated by high-throughput structural biology Stephen L. Gwaltney II, Kathleen Aertgeerts, Jun Feng, Stephen W. Kaldor, Daniel B. Kassel, Melinda Manuel, Marc Navre, G. Sridhar Prasad, Lihong Shi, Robert J. Skene, Jeffrey A. Stafford, Michael B. Wallace, Rongda Xu, Sheng Ye, Zhiyuan Zhang, David R. Webb | |
| 2:40 PM | 19 | Discovery of a potent CXCR2 receptor antagonist for the treatment of inflammatory disorders Michael P. Dwyer, Younong Yu, Jianping Chao, Cynthia Aki, Jianhua Chao, Biju Purakkattle, Diane Rindgen, Richard Bond, James Jakway, R. William Hipkin, James Fosetta, Waldemar Gonsiorek, Hong Bian, Jay Fine, J. Robert Merritt, Laura L. Rokosz, Bernd Kaiser, Ge Li, Wei Wang, Tara Stauffer, Lynne Ozgur, Arthur Taveras | |
| 3:15 PM | 20 | Discovery of AMG 131: A selective modulator of PPAR-γ Lawrence R. McGee, Steven M. Rubenstein, Jonathan B. Houze, Guosen Ye, Yang Li, R. Marc Learned, Jin-Long Chen, Zhulun Wang, Alykan Motani, Pieter B. Timmermans, Hisashi Shinkai, Atushi Hagiwara, Noburo Furukawa, Jun Nishiu, Motanao Nakamura | |
| 3:50 PM | 21 | Discovery of SCA-136, a novel 5-HT2C agonist, for the treatment of Schizophrenia P. Siva Ramamoorthy, Chad Beyer, Julie Brennan, John Dunlop, Stacey Gove, Steve Grauer, Boyd L. Harrison, Qian Lin, Jessica Malberg, Karen Marquis, Hossein Mazandarani, Mike Piesla, Claudine Pulicicchio, Sharon Rosenzwieg-Lipson, Ann-Marie Sabb, Lee Schechter, Gary Stack, Jean Zhang | |
| 4:25 PM | 22 | NVP-AEB071, an orally active inhibitor of early T cell activation for the prevention of graft rejection Jürgen Wagner, Rainer Albert, Nigel G. Cooke, Sylvain Cottens, Richard Sedrani, Maurice van Eis, Peter von Matt, Claus Ehrhardt, Jean-Pierre Evenou, Gerhard Zenke, Volker Brinkmann, Christian Beerli, Armin Brülisauer, Gisbert Weckbecker, Marc Bigaud, Charles Pally, Grazyna Wieczorek, Christoph Burkhart, Jianping Li, Barbara Nüsslein-Hildesheim, Christoph Heusser, Christian Bruns, Randall Morris, Gabriele Rummel, Wilhelm Stark, Gottfried Baier | |
Symposium Grid -- Division of Medicinal Chemistry -- Session Listing
Symposium Grid -- Drug Discovery -- Session Listing
The 231st ACS National Meeting, Atlanta, GA, March 26-30, 2006