ORGN 29 |
| 3,4-Dihydroquinolin-2(1H)-ones have potential biological and pharmacological significance. We have recently shown that enantiomerically pure benzothiazines can be synthesized via a completely selective, intramolecular addition of sulfoximine-stabilized carbanions to an α,β-unsaturated esters. We now present benzothiazines as templates for making a series of enatiomerically pure 3,4-dihydroquinolin-2(1H)-ones.
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Asymmetric Reactions and Syntheses
8:00 AM-11:40 AM, Sunday, 26 March 2006 Georgia World Congress Center -- C302, Oral
Division of Organic Chemistry |
