| MEDI | Wednesday, 31 August 2005 | ||
1:30 PM-4:30 PM Washington DC Convention Center -- Ballroom A, Oral | |||
MC4R Agonists and Antagonists | |||
| Organizer, Presiding: | R. P. Nargund | ||
| 1:30 PM | Introductory Remarks | ||
| 1:35 PM | 272 | Melanotropin ligands for the hMC4Rs: Multiple biological activities! One receptor? The challenge! Victor J. Hruby, Minying Cai, Jinfa Ying, Alexander Mayorov, Ravil Petrov, James Cain, Chad Park, Dev Trivedi | |
| 2:10 PM | 273 | Design of melanocortin receptor agonists by conformational restriction approach Xinrong Tian, Adrian G. Switzer, Rajesh K. Mishra, Timothy Field, Steve A. Derose, Eric Hu, Denny Denton, Nick Kim, Adam W. Mazur, Frank H. Ebetino, John A. Wos, Doreen Crossdoersen, Beth B. Pinney, Julie A. Farmer, Russell L. Sheldon, Martin E. Dowty, Cindy M. Obringer, Annyodile Colson | |
| 2:45 PM | 274 | Quinazolinone guanidines as MC4R agonists: SAR of unusual pharmacokinetic properties Jason D Speake | |
| 3:20 PM | 275 | Design and syntheses of human Melanocortin subtype-4 receptor (hMC4R) agonists: Discovery of the tert-butylpyrrolidine archetype Feroze Ujjainwalla | |
| 3:55 PM | 276 | Design, synthesis and characterization of potent and selective melanocortin-4 receptor antagonists Chen Chen | |
Symposium Grid -- Division of Medicinal Chemistry -- Session Listing
The 230th ACS National Meeting, in Washington, DC, Aug 28-Sept 1, 2005