MEDISunday, 13 March 2005

9:00 AM-12:20 PM Convention Center -- Room 6C, Oral
General Oral Session
Organizer:Daniel L. Flynn
Presiding:Brian S. J. Blagg
9:00 AMAllosteric enhancers of A1 adenosine receptors
Mahendra D. Chordia, Heidi Figler, Ray A. Olsson, Joel Linden
9:20 AMDiscovery and efficacy of the first orally administered derivatives of B-type natriuretic peptide
Kenneth D. James, Mark A. Miller, Navdeep B. Malkar, Diana Severynse-Stevens, Kevin G. Yarbrough, Karen Polowy, Mark J. Bednarcik, Robert E. Dugdell, Alessandro Cataliotti, John A. Schirger, Radha Krishnan, Monica E. Puskas, David Surguladze, Jenn L. Boyer, Nnochiri N. Ekwuribe, John C. Burnett Jr.
9:40 AMDesign and synthesis of orally efficacious Melanin Concentrating Hormone (MCH) receptor antagonists as antiobesity therapeutics
Mark D. McBriar, Henry Guzik, Ruo Xu, Jaroslava Paruchova, Shengjian Li, Anandan Palani, Sherry Shapiro, John W. Clader, William J. Greenlee, Brian E. Hawes, Hana Baker, Kim O'Neill, Brian Spar, Blair Weig
10:00 AMOver 100 peptide-activated GPCRs recognize turn motifs in ligands
David P. Fairlie, Joel D. A. Tyndall, Giovanni Abbenante, Bernhard Pfeiffer
10:20 AMNovel benzoxazocine analogues as potent analgesic agents
Andrew D. Baxter, Michael Lyne, Stuart Brown
10:40 AMOpioid Receptor Like (ORL1/NOP) agonists as novel analgesics
Paul D Ratcliffe
11:00 AMA chemical genetics approach for the discovery of novel anti-cancer agents and targets: Identification of transferrin receptor as the molecular target of gambogic acid, a rapid and potent apoptosis-inducer
Sui Xiong Cai, Han-Zhong Zhang, Katayoun Jessen, Sergei Maliartchouk, Jean Yu Wang, Nicki English, Ling Qiu, Nilantha Sirisoma, Songchun Jiang, Jared Kuemerle, John Drewe, Kurt Gehlsen, Ben Tseng, Shailaja Kasibhatla
11:20 AMA chemogenomic approach for ion channel and transport modulators
Holger Heitsch
11:40 AMClofibrate-induced changes in the lipid metabolome
Craig E. Wheelock, John W. Newman, Steven M. Watkins, Bruce D. Hammock
12:00 PMRational design of multiple ligands: Risks and benefits
J. Richard Morphy

Symposium Grid -- Division of Medicinal Chemistry -- Session Listing

The 229th ACS National Meeting, in San Diego, CA, March 13-17, 2005