ORGNThursday, August 26, 2004

1:00 PM-5:00 PM Pennsylvania Convention Center -- 202B, Oral
Combinatorial, Parallel, and Solid-Phase Chemistry
Presiding:Roland E. Dolle
1:00 PM Solid/solution Phase Annulation (SPAnTM) technology: Single–step derivatization of primary amines to heterocycles
Roland E. Dolle, Blanca Martinez-Teipel, Calum MacLeod
1:20 PM Tungsten alkyne-ol cyclizations with aldehydes to form biologically interesting molecules
Allen S. Kesselring, Scott R. Gilbertson
1:40 PM DendriGels as new high-loading hybrid materials for multistep synthesis of drug-analogues
Rainer Haag, Sebastian Roller, Holger Türk
2:00 PM Novel MCR 3 reaction leading to an interesting zwitterionic structure: Parallel synthesis of pyridinium-pyrazol-3-olate inner salts
László Ürge, László Varga, Tamás Nagy, György Dormán, Ferenc Kálmán, Ferenc Darvas
2:20 PM Preparation of bicyclic reverse turn for Leu-enkephalin analogues
Xuyuan Gu, Jinfa Ying, Jimes P. Cain, Byoung Min, Victor J. Hruby
2:40 PM P1-site diversity in peptide isostere libraries via smooth CC-couplings on linker reagents
Jörg Rademann
3:00 PM Second generation C-linked AFGP analogues : Tailoring recrystallization-inhibition and thermal hysteresis properties
Vincent R. Bouvet, Anastasia V. Murphy, Matthew F. L. Parker, Robert N. Ben
3:20 PM Pseudo-dynamic combinatorial chemistry: A new receptor-assisted combinatorial method for identifying enzyme inhibitors
Jeremy D. Cheeseman, Andrew D Corbett, David Soriano del Amo, Romas J. Kazlauskas, James L. Gleason
3:40 PM Simple and effective tagging system for solution phase synthesis
Jordan Blodgett, Tingyu Li
4:00 PM Polymer-supported metal scavengers and their applications in modern synthesis
Paul A Boguszewski, Andrew F Coffey, John W Davies, Alasdair A MacDonald, Aubrey J Mendonca, Frank P Warner
4:20 PM Light-directed combinatorial chemistry
Peter J. Belshaw, Alex Shaginian, Shane T. Flickinger, Madhusudan Patel
4:40 PM Robotic-assisted synthesis optimization of benzylphophonic acid using six-sigma quality methods
David B. Engel, Donald W. Whisenhunt Jr.

Symposium Grid -- Division of Organic Chemistry -- Session Listing

The 228th ACS National Meeting, in Philadelphia, PA, August 22-26, 2004