Mechanistic studies of Scholl cascade reactions

ORGN 238

Pawel Rempala, Jiri Kroulik, and Benjamin T. King. Department of Chemistry, University of Nevada, Reno, NV 89557
The Scholl reaction was investigated at the B3LYP/6-31G(d) level of theory for the conversion of a series of 1,2,...,n-polyphenylbenzenes (n = 3, 4, 6) to the corresponding planar polycyclic aromatic hydrocarbons. The formation of C-C bonds is stepwise, with a repetitive sequence of protonation, intramolecular electrophilic C-C bond formation, deprotonation, and oxidative dehydrogenation. An alternative mechanism involving the initial formation of a radical cation is unlikely due to high C-C bond formation barriers. The formation of the first C-C bond is rate determining, accounting for the ease of cascade Scholl condensations. The occasionally observed accumulation of intermediates is an electrochemical phenomenon.