ORGN 123 |
| William R. Perrault, Paul M. Herrinton, Richard A. Hohler, Joseph W. Strohbach, Steven P. Tanis, and Malcolm W. Moon. Early Process Research and Development, Pharmacia, 7000 Portage Rd., Kalamazoo, MI 49004 |
| A scalable route to a pyridoquinoxaline antiviral compound was developed which allowed for the rapid preparation of significant quantities of material to support development needs. A method of preparing the key heterocyclic ring was developed which involved a one step cyclization/ deacylation procedure. |
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New Reactions and Methodology, Metal-Mediated Reactions, Heterocycles and Aromatics
8:00 PM-10:00 PM, Sunday, March 28, 2004 Anaheim Convention Center -- Hall A, Poster
Division of Organic Chemistry |