| ORGN | Sunday, September 7, 2003 | ||
1:00 PM-5:00 PM Sheraton New York -- Royal Ballroom B,Oral | |||
Process R&D | |||
| Presiding: | J. Christopher McWilliams | ||
| 1:00 PM | 73 | Practical synthesis of the new carbapenem antibiotic ertapenem sodium J. M. Williams, K. M. J. Brands, K. M. Conrad, B. Pipik, K. A. Savary, F-R. Tsay, P. G. Houghton, R. T. Skerlj, R. B. Jobson, G. Marchesini, L. M. DiMichele, U-H. Dolling | |
| 1:20 PM | 74 | Enantio- and regioselective opening of 2-alkyl nosylaziridines by indoles mediated by boron trifluoride. Application to a practical synthesis of a GnRH antagonist Roger N. Farr, Ramon J. Alabaster, John Y. L. Chung, Bridgette Craig, John S. Edwards, Andrew W. Gibson, Guo-Jie Ho, Guy R. Humphrey, Simon A. Johnson, Edward J. J. Grabowski | |
| 1:40 PM | 75 | A general approach to 2-substituted indoles Jacqueline H. Smitrovich, Chuanxing Qu, Ian W. Davies, Dave Hughes | |
| 2:00 PM | 76 | Process development in the preparation of substituted oxazoles Kenneth J. Natalie, Andrew Rusowicz, Dale J. Vanyo, Raymond E. Weaver, Ambarish K. Singh | |
| 2:20 PM | 77 | Practical synthesis of a 5-aryl-1,3-thiazolidine-2,4-dione PPAR agonist Michael H. Kress, M. David Weingarten, Christopher J. Welch, Maria Beconi, David J. Mathre, James M. McNamara | |
| 2:40 PM | 78 | Synthesis of a dual PPAR agonist and the formation of a sterically congested alpha-aryloxyisobutyric acid Raymond J. Cvetovich, John Y. L. Chung, Michael H. Kress, Joseph S. Amato, George Zhou, Louis Matty, F.R. Tsay, Zhen Li | |
| 3:00 PM | 79 | Development of the synthesis of BMS-250749, a potent topoisomerase inhibitor Jianji Wang, Miguel Rosigana, Daniel Watson, Eric Dowdy, Meena Rao, Robert Discordia, Nachimuthu Soundarajan, Wen-Sen Li | |
| 3:20 PM | 80 | Chromatography in support of pharmaceutical process research Christopher J. Welch | |
| 3:40 PM | 81 | A convenient one-pot synthesis of 1,8-naphthyridones Shawn A. Springfield, Karen Marcantonio, Scott Ceglia, Jennifer Albaneze-Walker, Peter G. Dormer, Todd D. Nelson, Jerry A. Murry | |
| 4:00 PM | 82 | Practical process solutions for Suzuki coupling reactions Atul S. Kotnis, Kenneth J. Natalie, Bruce Lotz, Ambarish K. Singh, Raymond E. Weaver, David Kascur, David Thurston, Keming Zhu, J. Siva Prasad | |
| 4:20 PM | 83 | Palladium mediated Ferrier rearrangement type glycosidation with aromatization prone xylo-furanoid glycals for the synthesis of biologically active nucleosides Anusuya Choudhury, Michael E. Pierce, Dieu Nguyen, Louis Storace, Pat Confalone | |
| 4:40 PM | 84 | Synthesis of an alpha-alkylamino pyrazinone thrombin inhibitor mediated by 2-pyridylthioimidate-ZnCl2 complexes Raymond J. Cvetovich, John Y. L. Chung, Fuh-Rong Tsay, Peter G. Dormer, Lisa DiMichele, Bing Mao, Robert Wenslow | |
Symposium Grid -- Division of Organic Chemistry -- Session Listing
The 226th ACS National Meeting, New York, NY, September 7-11, 2003