| ORGN | Sunday, September 7, 2003 | ||
8:00 PM-10:00 PM Hilton New York -- Rhinelander Center,Poster | |||
Methodology, Process R&D, Combinatorial, Total Synthesis | |||
| Organizer: | L. McElwee-White | 85 | Activation of kenner's N-Acyl sulfonamide "safety-catch" linker using Pd(0)-catalyzed allylation Yi He, Laura L. Kiessling |
86 | Applications of organometallic chemistry in the pharmaceutical industry: A mechanistic and kinetic study of the MK-869 hydrogenation network Thorsten Rosner, Shane Krska, Karel M.J. Brands, Karen M. Conrad, Fuh-Rong Tsay, Fred W. Hartner, Edward G. Corley, Robert A. Reamer, Robert D. Larsen, Mahmoud Kaba, Yongkui Sun |
87 | Asymmetric synthesis of 3-aminohexose glycals: a 7-step synthesis of a protected vancosamine glycal Wonsuk Chang, Kathlyn A. Parker |
88 | Directional bromination of xylenes Kaitao Lu, Der-Haw Wang, Peter C. Zhu |
89 | Novel applications of Biginelli reaction. Solution phase parallel synthesis of dihydropyrimidinone, dihydropyrimidinthione, dihydropyrimidothiazine libraries András Lukács, László Ürge, György Dormán, Ferenc Kálmán, Ferenc Darvas |
90 | Studies toward the total synthesis of Plakevulin A Katherine L. Hervert, Louis S. Hegedus |
91 | Synthesis of a novel monomer bis(p-hydroxyphenyl)bis(p-chlorophenyl)methane with a tetrahedral configuration Guodong Dang, Wanjin Zhang, Y. Wei |
92 | Synthesis of macrocyclic a-ketoamides via ring-closing metathesis John T. Randolph, Peggy Huang, Larry Klein, Dale Kempf |
93 | Total synthesis of molluscan polypropionates using a novel Lewis acid catalyzed cyclization Aubry Miller, Dirk Trauner |
94 | Towards the total synthesis of the anticancer agent Roseophilin E.M.E. Viseux, P.J.P. Parsons, J.B.J. Pavey |
95 | Two complementary approaches on 2-alkoxy carboxylic acid synthesis from 1,3-dioxolan-4-ones Leonard L. Winneroski Jr., Yanping Xu |
96 | Weinreb amide functionalized dipolar species Richard.W Franck, Ajit Kumar Parhi |
97 | Synthesis of 2,3-disubstituted benzo[b]furans by the palladium-catalyzed coupling of o-iodoanisole and terminal alkynes, followed by electrophilic cyclization Dawei Yue, Richard C Larock |
98 | Synthesis and reactivity of allenamides and ynamides Michael R. Tracey, Richard Hsung |
99 | Stereoselective pericyclic reactions involving ynamides Richard Hsung, Jason A. Mulder, Mike O. Frederick, Michael R. Tracey, Craig A. Zificsak, Robert H. Lambeth III |
100 | Formal [3+3] cycloaddition strategy towards synthesis of highly functionalized piperidines Nadiya Sydorenko, Richard Hsung, Juliet M. Hahn, Ossama S. Darwish |
101 | Room temperature ionic liquids from a biorenewable resource - D-Fructose Maurice Okello, Scott T Handy |
102 | Solvent dependent reactions of benzylsulfonylacetic acids N. Srinivasa Reddy, E. Premkumar Reddy, M.V. Ramana Reddy |
103 | Studies toward an enantioselective total synthesis of tremulenediol A and tremulenolide A: development of a highly regioselective Rh(I)-catalyzed allylic alkylation reaction Brandon L. Ashfeld, Stephen F. Martin |
104 | Practical route to -ß-alkylated-1,3,2-oxazaborolidines via BH substitution Margarita Ortiz-Marciales, Eduvigis Gonzalez, Melvin De Jesus, Sandraliz Espinosa, Wildeliz Correa |
105 | Reactions of hydrazine with a-cyanocinnamate esters: an unexpected fragmentation Paul J. Erdman, David E. Lewis |
106 | Convenient one-pot synthesis of dihydroquinolones Glen C. Gullickson, David E. Lewis |
107 | One-pot synthesis of N-substituted phthalimides from methylarenes Saliya de Silva, Saurabh Dhruve, David Isidor, Magambo Nyakirang’ani, Supun Pathirana, Edinam Klu, Tope Osinaiya |
108 | Oxocarbenium ion cyclizations for the synthesis of fumagillin analogues Fatoumata Camara, Johana Angarita, Galyna Pushchinska, David R. Mootoo |
109 | New reagents for asymmetric electrophilic amination Alan Armstrong, Ian E. Edmonds, Martin Swarbrick |
110 | New N- and O-arylations with potassium aryltrifluoroborates and cupric acetate Christopher W. Ajello, Bertrand Le Bourdonnec, Roland E. Dolle |
111 | Highly efficient and chemoselective synthesis of 3, 5-diketoesters by Lipase catalyzed transesterification: application in resolution of racemic alcohols and desymmetrization of meso diols A. Ian Scott, Samik Nanda |
112 | Highly efficient synthesis of azabicyclo[X.Y.0]alkane amino acids by Rh-catalyzed cyclohydrocarbonylation Wen-Hua Chiou, Nobuhiro Mizutani, Iwao Ojima |
113 | Isoureas: versatile synthetic intermediates Bruno Linclau, Stefano Crosignani, Zhengning Li, Patrick Lecarpentier |
114 | Mild and efficient conversion of formamides to isocyanides using the complex of 2,4,6-trichloro[1,3,5]triazine and N,N-dimethyl formamide Hagyoung Lee, Ki-Jong Han, Misoo Kim |
115 | Diastereoselective synthesis of 2,6-cis-disubstituted tetrahydopyranones: Studies toward the enantioselective preparation of tetrahydropyranone natural products Christopher A. Lee, Paul E. Floreancig |
116 | Efficient amination of sulfides with a ketomalonate derived oxaziridine Alan Armstrong, Richard S. Cooke |
117 | Efficient synthesis of 2-alkyl-2-phenoxypropionic acids via a-lactone pathway Jeremy York, Leonard L. Winneroski Jr., Yanping Xu |
118 | Development of a general strategy for the stereoselective synthesis of highly functionalized carbocycles via an enolate Claisen/diastereoselective ring-closing metathesis protocol John Robinson, Anthony D. Piscopio |
119 | Development of a novel three component coupling process: Synthesis of substituted pyrimidinones Dengming Xiao, Eugene Tarlton, Kevin Koch, Anthony D. Piscopio |
120 | CsOH-promoted epoxide ring-opening with phosphines: Mild and efficient synthesis of monohydroxyphosphines Ashlee A. Robinson, Brandon Frank, Daniel L. Fox, Ralph Nicholas Salvatore |
121 | Convenient procedure for the formylation of amines using formic acid and bis(trichloromethyl) carbonate Misoo Kim, Ki-Jong Han, Hagyoung Lee |
122 | Desymmetrising aza-wittig reactions Stephen P Marsden, Jenna Jamal, M. Jonathan Fray |
123 | b-Hydroxy nitriles and 1,3-amino alcohols from epoxides: Improved, one-pot procedures using LiCN in THF James A. Ciaccio, Michael Smrtka, William Maio |
124 | A new methylenecyclopentane annulation process H.J. Liu, Liang-Rern Kung, Che-Hao Tu |
125 | A novel route to azobenzenes and its application towards synthesis of dendritic and cyclic polyazobenzenes Cheon-Gyu Cho, Young-Kwan Lim, Kang-Sang Lee |
126 | Arylchloride-organoboron coupling with bulky imidazolium-palladium carbene catalysts Merritt B. Andrus, Chun Song, Yudao Ma, Wei Jiang |
127 | A scaleable synthesis of 2,4-disubstituted imidazoles by condensation of amidines and a-haloketones Z. Bryan Li, Charles K-F Chiu, Richard F. Hank, Jerry Murry, Joshua Roth, Harry Tobiassen |
128 | Group selective intramolecular cycloadditions of sulfenic acids to prochiral alkenes Patrizia Tisselli, Richard S. Grainger |
129 | Preparation of pivaloyl hydrazide in water Z. Bryan Li, Raymond J. Bemish, David R. Bill, Steven Brenek, Richard A. Buzon, Charles K-F. Chiu, Lisa Newell |
130 | MgI2 catalyze the aldol-type reaction: a general route to synthesis of (E)-ß-iodovinyl-ß'-hydroxyketones Han-Xun Wei, Hui Hu, Mohamed A Farag, Paul W. Pare |
131 | Radical-induced cyclopentannulation using nitroaldol(Henry)-derived intermediates Frederick A. Luzzio, Joel P. Ott |
132 | An improved synthetic route to analogues of the new SERMs WAY-138923 and WAY-140424 Arthur A. Santilli, Marci C. Koko, Andrew Q. Viet |
133 | Synthesis of (S,S)-2-(2-morpholin-2-yl-2-phenyl-methoxy)-phenol Jaya Prabhakaran, Vattoly J Majo, Theodore S. Wang, J. John Mann, J. S. Dileep Kumar |
134 | Microwave assisted multi-component reactions Heather Tye, Mark Whittaker, Sarah M Ireland |
135 | Organic reactions in water using hydrophobic polymer-supported Brfnsted acid catalysts Shinya Iimura, Daisuke Nobutou, Kei Manabe, Shu Kobayashi |
136 | An investigation of the zinc organometallic intermediate in the syn-selective tandem chain extension-aldol reaction of ß-keto esters Karelle S. Aiken, Charles K. Zercher, Su-jen Lai |
137 | Diastereoselective alkylations of beta-tetrazolyl propionic acids Michael G. Yang, Dilip P. Modi, Wayne F. Rankin, Jianliang Shi, Ruth R. Wexler, Richard E. Olson |
138 | Dimethyldioxirane mediated rearrangement of bicyclic imidazoles Yong He, Hongwang Du, Carl J. Lovely |
139 | Side chain incorporation in ketomethylene isosteres Weimin Lin, Nancy Tryder, Fan Su, Charles K. Zercher |
140 | Regioselectivity in Stille coupling reactions of 3,5-dibromo-2-pyrone Cheon-Gyu Cho, Won-Suk Kim |
141 | Novel reaction of propargyl alcohols with alkynes promoted by boron trihalides and titanium tetrahalides: synthesis of halogenated 1,4-enynes George W Kabalka, Zhongzhi Wu, Yuhong Ju |
142 | Practical routes for the synthesis of b,g-unsaturated amino acids Stephen P Marsden, Paul Alexander, John C. Reader |
143 | Facile synthesis of substituted 2-(amidoalkyl)azoles Dennis J. Hlasta, Craig A. Zificsak |
144 | A practical synthesis of 2,4-disubstituted resorcinol derivatives Scott S. Ceglia, Michael H. Kress, James M. McNamara |
145 | Efficient synthesis of 1,4-diaminophthalazines, an important moiety of E8010, a novel PDE type 5 inhibitor Kazuhiro Yoshizawa, Shinya Abe, Yuki Komatsu, Ken Furukawa, Naoyuki Shimomura |
146 | Intramolecular allylation of erythromycin derivatives Su Yu, Xiu Wang, Ashok V. Bhatia |
147 | Mechanistic insight into a highly selective preparation of imidazo[1,2-a]pyrimidine Yun Qian, Michael Breslav, Rosie Chang, Helen Chao, Rong Feng, Steven Goltra, Jeffrey Grimm, Mark Haslego, Aihua Huang, Sergio Cesco-Cancian, Charles Shaw, Cynthia Maryanoff, Mitul Patel, Kirk L. Sorgi, James Weber, Xinzhen(Jane) Xiang, Dawei Xu |
148 | Optimization of a process for the preparation of the farnesyl transferase inhibitor BMS-214662 Zhenrong Guo, Boguslaw M. Mudryk, Zhinong Gao, Terence Moore, Cary McConlogue, David Kronenthal, Melanie Miller, Chien-Kuang Chen |
149 | Stereoselective cyclizations of donor-acceptor cyclopropanes Brian L. Pagenkopf, Ming Yu |
150 | New linkers for traceless cleavage strategies in solid phase synthesis Jun Guo, Peter J. H. Scott, Patrick G Steel, Ian B. Campbell |
151 | The development of high-load, soluble reagents via ROMP: Oligomeric sulfoxides and benzyl sulfonates Mianji Zhang, Joel D. Moore, Daniel L. Flynn, Paul R. Hanson |
152 | Capture-ROMP-release: Applications in synthesis Shubhasish Mukherjee, Andrew M. Harned, Kevin W. C. Poon, Daniel L. Flynn, Paul R. Hanson |
153 | Novel orthogonal strategy toward solid phase synthesis of 1,3,5-substituted triazines Jae Wook Lee, Jacqueline T. Bork, Sonya M. Khersonsky, Young-Tae Chang |
154 | Tubuyzine: Novel anti-microtubule compound from triazine-libraries Daniel P. Walsh, Sonya M. Khersonsky, Young-Tae Chang |
155 | On column clean synthesis of an array of benzofurans using silica-supported reagents cartridges Shahnaz Ghassemi, P. C. Rahn |
156 | Progress towards a diversity-oriented synthesis of linear polyketides Daniel E. Macks, James M. Rogér, Derek S. Tan |
157 | Selective catch and release of a synthetically useful phosphine Jennifer L. Marugg, Martin L. Neitzel, John Tucker |
158 | Novel and efficient method for solution phase parallel synthesis of amides from acid chlorides and amines using PS-HOBT Nand Baindur, Naresh Chadha, Mark R. Player |
159 | Polymer-supported toluenesulfonic acid: A versatile tool for expedient purification or scavenging of amines and nitrogen heterocycles Owen W. Gooding, Jeff W. Labadie, Sukanta Bhattacharyya, Tejal Parekh, Lanchi Vo |
160 | Solid phase synthesis of fluorescent Ras-mimetic lipopeptides: Novel cell-permeable substrates of protein palmitoyl acyltransferase Sangarappan Sivakumar, Steffen P. Creaser, Blake R. Peterson |
161 | Spacer-modified diol-functionalised polystyrene resins: Synthesis and applications Toby B. Reeve, Sandeep Handa, Philip W.D. Dyer |
162 | Stereoselective diversity-oriented synthesis of spiroketals Justin S. Potuzak, Sirkka B. Moilanen, Derek S. Tan |
163 | Towards supported olefin-metathesis catalysts Samuel Suhard, Philip W.D. Dyer |
164 | An efficient capping residual hydroxythiophenol on solid support for synthesis of high quality compound library Luyong Jiang, Alex Chucholowski, Rongshi Li |
165 | An efficient synthesis of a bicyclic gamma-lactam library on solid support Tong Zhu, Zheng Yan, Rongshi Li |
166 | Expanded stereochemical diversity in the diversity-oriented synthesis of spiroketals Sirkka B. Moilanen, Justin S. Potuzak, Derek S. Tan |
167 | Paper Withdrawn | 168 | Development of pseudoephedrine chiral linkers for asymmetric alkylations on solid phase Panee C. Hutchison, Tom D. Heightman, David J. Procter |
169 | Traceless solid phase synthesis of substituted benzoimidazolones Wen-Ren Li, Chih-Chung Wang |
170 | Solid-phase oligosaccharide synthesis with real-time reaction monitoring by color test Shino Manabe, Yukishige Ito |
171 | New Holliday Junction inhibitors and Class B synergimycin derivatives Irene Medina, Enrique V. Azevedo, Shelli R McAlpine |
172 | Novel Quinopristin antibiotics: Structural derivatives Chris Carroll, Jennifer L. Robinson, Shelli R McAlpine |
173 | Novel antibiotics: Class B synergimycin derivatives and site specific recombination inhibitors Maggie J. Shale, Lisa A. Liotta, Megan L Bolla, Shelli R McAlpine |
174 | Synthesis of enantiomerically pure tetrahydrofurans using ylides: Application to the total synthesis of haterumalide NA Jennifer Schomaker, Pulgam Veera Reddy, Babak Borhan |
175 | Synthetic studies toward (-)-galanthamine. Beckmann rearrangement approach for the seven-membered ring Keith R. Buszek |
176 | Synthetic studies toward dregeanin. Facile construction of the saturated eight-membered lactone ring Keith R. Buszek |
177 | Synthetic studies towards Isaindigotidione and its analogues Ch Yan Poon, Pauline Chiu |
178 | The first enantioselective synthesis of hexahydro TMC-69: A novel method for the construction of 5,6-disubstituted dihydropyran-3-nones Dengming Xiao, Anthony D. Piscopio |
179 | Total synthesis of azaspiracid. Construction of the CDE ring system Keith R. Buszek, Tony S. Gibson, Brian C. Reinhardt, Jason R. Sunde |
180 | Total synthesis of the sesquiterpenoid copaene Sasan Karimi, Julia Christodoulou |
181 | Towards the new diazonamide A: Synthesis of a tyrosine-derived benzofuranone Francine N Palmer, Christopher J Moody |
182 | Studies towards the total synthesis of FR182877 Frederick W. Goldberg, Alan Armstrong, David Sandham |
183 | Synthesis of (+)-decarestrictine L and the C17-C24 fragment of ambruticin via C-glycosidation Julie M. Lukesh, William A. Donaldson |
184 | Synthesis of M3 and M1 metabolites of HIV protease inhibitor Nelfinavir Mesylate Aniruddha P. Patwardhan, Mitali Ghoshal, Jason Klein, Christa Hubner-Parajsz, Josef Endl, Sigrun Metz, Angela Puhlmann, Gerald Sigler, Jane Tsai, Joseph Passarelli |
185 | Synthetic efforts towards Amphidinolide T1 Benjamin R. Travis, Babak Borhan |
186 | Studies toward the total synthesis of bryostatin 1 Gary E. Keck, Anh P. Truong |
187 | Studies toward the total synthesis of halichlorine Gary E. Keck, Stacey A. Dalton |
188 | Studies toward the total synthesis of swinholide A Gary E. Keck, Lars Heumann |
189 | Studies toward the total synthesis of epothilone b Gary E. Keck, Robert L. Giles |
190 | Progress toward the synthesis of Arisugacins and Territrems Michael E. Jung, Sun-Joon Min |
191 | Progress toward the total synthesis of pseudolaric acids Zhe Geng, Pauline Chiu |
192 | Paper Withdrawn | 193 | Studies directed toward the total synthesis of gigantecin Jin She, Michael T. Crimmins |
194 | Exploiting olefin metathesis for the construction of the core of SCH 351448 Michael T. Crimmins, Grace R. Smalley |
195 | Studies toward synthesis of polycyclic polyprenylated acylphloroglucinols Robert B. Grossman, Roxana Ciochina |
196 | Studies directed towards total synthesis of Rhododaurichromanic acid A Aleksey V. Kurdyumov, Kristen M. Ihlen, Jiashi Wang, Richard P. Hsung |
197 | Studies directed towards a total synthesis of pinnaic acid Rameshkumar Chellappan, Richard Hsung |
198 | New approaches to the 13C labelling of (+)-catechin Neil D. Forrest, Richard C. Hartley, Alan Crozier |
199 | Catalytic asymmetric synthesis of the chiral tetraene acyl side chain of papulacandin D Huanyan Cao, Kathlyn A. Parker |
200 | Progress on the total synthesis of SNF4435C and D Yeon-Hee Lim, Kathlyn A. Parker |
201 | Asymmetric total synthesis of C-glycoside of alpha-galactosylceramide Jun Pu, Richard W. Franck |
202 | Studies towards the total synthesis of the marine alkaloid sarain A Sungwoo Hong, Steven M. Weinreb |
203 | Total synthesis of C-glycosides of isoflavone Vishnu Vardhan Reddy Karnati, Wu-Yan Zhang, David Y.W. Lee |
204 | Studies toward the total synthesis of lamellarins Yanan Zhang, Scott T Handy, Jennifer M Lewis, Jesse J Sabatini |
205 | Synthetic studies of himbacine and its congeners featuring intermolecular Diels-Alder reaction Masanori Takadoi, Tomoyuki Kawai, Kentaro Yamaguchi, Shiro Terashima |
206 | Utilization of hidden meso-symmetry towards the synthesis of the C22-C36 segment of halichondrin B Valerie A. Keller, Steven D. Burke |
207 | Total synthesis of a conjugate of a NAALADase inhibitor Pingyu Ding, Paul Helquist, Marvin J. Miller |
208 | Progress toward the total synthesis of reticulidin A and deoxyreticulidin A Jacob I. Wasserman, Michael E. Jung |
209 | Synthesis of allylphosphinoyl phenylsulfone: a conjunctive reagent for synthesis of conjugated dienes Xiaojin Li, Philip L. Fuchs |
Symposium Grid -- Division of Organic Chemistry -- Session Listing
The 226th ACS National Meeting, New York, NY, September 7-11, 2003