| ORGN | Wednesday, September 10, 2003 | ||
8:30 AM-11:25 AM Sheraton New York -- Imperial Ballroom A,Oral | |||
Technical Achievement in Organic Chemistry Awards | |||
| Organizer, Presiding: | William J. Greenlee | ||
| 8:30 AM | 471 | Process development of PPAR-gamma dominant agonist LY519818 John R. Rizzo, Tony Y. Zhang, Samuel R. Wendel, Chauncey D. Jones, Robert W. Towsley | |
| 8:55 AM | 472 | Development of novel series of potent phosphodiesterase-4 (PDE4) inhibitors: SAR studies on substituted 4-(2,2-diarylethyl)pyridine-N-oxides Richard Frenette | |
| 9:20 AM | 473 | TIBO to TMC-125: the discovery of potent and broad spectrum anti-HIV NNRTIs Donald W. Ludovici, Michael J. Kukla, Barte L. De Corte, Robert W. Kavash, Chih Y. Ho, Hong Ye, Mark A. Lichtenstein, Philip P. Grous, Suma Krishnan, Henry J. Breslin, Winston Ho, Malolm K. Scott, James D. Rodgers, Richard Mohrbacher, Craig J. Diamond, Milton Miranda, Cynthia L. Fedde, Ronald G. Sherrill, T. Kevin Hitchens, Koen Andries, Marie-Pierre de Béthune, Hilde Azijn, Henry E. L. Moereels, Lucien M.H. Koymans, Marc R. de Jonge, Koen J.A. Van Aken, Frederik F.D. Daeyaert, Paul Lewi, Kalyan Das, Edward Arnold, Erik De Clercq, Rudi Pauwels, Jan Heeres, Paul A. J. Janssen | |
| 9:45 AM | 474 | Synthesis and SAR of 3(2H)-pyridazinones as selective COX-2 inhibitors: Discovery of ABT-963 Lawrence A. Black, R. Athalye, Anwer Basha, Pramila A. Bhatia, Jennifer J. Bouska, Linda Chernesky, John DeMattei, Todd Gane, Ahmed Hakeem, Richard Harris, Cathy Henry, Peer B Jacobson, Jianguo Ji, Teodozyj Kolasa, Michael E. Kort, Daniel Larson, Huaqing Liu, Sandy Majest, Kennan Marsh, Catherine M. McCarty, Merrill Nuss, Meena V. Patel, Daisy Pireh, Marina Pliuschev, James Ratajczyk, Jeffrey J. Rohde, Teresa Rosenberg, Richard J. Sciotti, S. Surapaneni, Frank L. Wagenaar, Michael R. Michaelides, Andrew O. Stewart, Michael J. Coghlan, James Summers, Clint D. W. Brooks, George W. Carter, Randy L. Bell | |
| 10:10 AM | 475 | Efficiency, robustness, and environmental responsibility: Technical process chemistry in a pharmaceutical setting John Tucker | |
| 10:35 AM | 476 | Butynyl ether derivatives as inhibitors of TACE Mila Du | |
| 11:00 AM | 477 | Synthesis of novel benzazepine oxazolidinone antibacterials Paul Johnson | |
Technical Achievement in Organic Chemistry Awards -- Next Session
Symposium Grid -- Division of Organic Chemistry -- Session Listing
The 226th ACS National Meeting, New York, NY, September 7-11, 2003