| ORGN | Sunday, March 23, 2003 | ||
8:00 PM-10:00 PM Convention Center -- Hall G,Poster | |||
Molecular Recognition, Combinatorial, Bioorganic | |||
| Organizer: | L. McElwee-White | 61 | Application of a flexible, asymmetric synthesis of (5R)-thiolactomycin to develop new inhibitors of type I fatty acid synthase Jill M. McFadden, Susan M. Medghalchi, Jagan N. Thupari, Michael L. Pinn, Aravinda Vadlamudi, Katherine I. Miller, Francis P. Kuhajda, Craig A. Townsend |
62 | Substrate specificity of b-lactam synthetase Fumitaka Kudo, Craig A. Townsend |
63 | Synthesis and diffusion measurements of flexible tetraether acyclic bisphosphocholines Wilma Febo-Ayala, Scott A. Bradley, Aniruddha Patwardhan, David H. Thompson |
64 | Synthesis of a thionated inhibitor for thimet oligopeptidase Samantha J. Friedman, Julia H Miwa |
65 | Synthesis of naturally occurring lipids and derivatives Jin-Young Yoon, Jin-Seon Park, Mi-Geum Kim, Young-Ah Kim, So-Yeop Han |
66 | Total synthesis of mauritine D, amphibine E, and their epimers Young-Ah Kim, Hae-Jeong Min, So-Yeop Han |
67 | A novel synthesis of peptidomimetics based on a pyridone scaffold: A versatile three-component reaction Namal C Warshakoon, Rodney D. Bush |
68 | Construction of a chemical library of unnatural polyketides by plant polyketide synthases Ikuro Abe, Hiroyuki Morita, Yusuke Takahashi, Hiroshi Noguchi |
69 | Synthesis of cyclic thiooligosaccharides: b-1,6-thio-linked cycloglucopyranosides Linfeng Fan, Ole Hindsgaul |
70 | Thermodynamics of reversibly formed encapsulation complexes Elke C. Ullrich, Julius Rebek |
71 | Triply interlocked 2-D self-assembly of modified triphenylenes Carsten Siering, Roland Fröhlich, Siegfried R. Waldvogel |
72 | Synthesis of D-leucine derived PNA monomers: DiSC2(5) aggregate formation on modified PNA/DNA templates Rojendra Singh, Isil Dilek, Bruce Armitage |
73 | Effect of template length on the formation of cyanine dye aggregates on PNA-DNA duplexes Violeta L. Marin, Bruce Armitage |
74 | Synthesis of new pyrene-containing, metal-chelating lipids and sensing of cupric ions Bidhan C Roy, Binita Chandra, Daniel Hromas, Sanku Mallik |
75 | Paper Withdrawn | 76 | A new electron acceptor for supramolecular chemistry Kathryn A. McMenimen, Joseph B. Carroll, Vincent M. Rotello, Thibaut Jarrosson, Darren G. Hamilton |
77 | Surface-functionalized dendritic architectures Pandi Bharathi, D Vutukuri, S Thayumanavan |
78 | Water-soluble calix[4]arenes for molecular recognition and encapsulation Suazette N. Reid, Suzanne B. Shuker |
79 | Progress toward a synthesis of a half-chloptosin cyclohexapeptide Jee-Youn Lee, Young-Ah Kim, So-Yeop Han |
80 | Small catalytic peptides that operate an enamine mechanism: Improvement of catalytic activity and substrate specificity Fujie Tanaka, Roberta Fuller, Carlos F. Barbas III |
81 | Convergent evolution of aldolase antibodies in vitro: Correlation between catalytic activity and diketone binding within a set of aldolase antibodies Fujie Tanaka, Roberta Fuller, Hyunbo Shim, Marikka Elia, Richard A. Lerner, Carlos F. Barbas III |
82 | Polyhedral oligomeric silsequioxane-based supramolecular assemblies Joseph B. Carroll, Vincent M. Rotello |
83 | Porphyrin-appended anion receptors Stephen D. Starnes, Sailaja Arungundram, Colene H. Saunders, Jeff C. Harper |
84 | Sequence-selective enhancement of guanine alkylation by a minor groove binder Sridhar Varadarajan, Barry Gold |
85 | Sequence-specific DNA methylation in the minor groove Sridhar Varadarajan, Dharini Shah, Prasad Dande, Samuel Settles, Barry Gold |
86 | Molecular assembly of 1,2- and 1,3-bis(cyanomethyl)benzene with silver salts Gerardo Marquez, Douglas M. Ho, Kathleen V. Kilway |
87 | Molecular assembly of polycyanovinylarenes with silver salts John R. VanScoy, Douglas M. Ho, Kathleen V. Kilway |
88 | Molecular recognition of nucleic acids through SELEX Joseph C. Manimala, Andrew D. Ellington, Eric V. Anslyn |
89 | Origins of selectivity in noncovalent molecular imprinted polymers Ryan L. Simon, Jason N. Campbell, David A. Spivak |
90 | Synthesis and characterization of a novel L-serine-based cross-linking monomer for molecular imprinting Martha Sibrian-Vazquez, David A. Spivak |
91 | Influences on MIP selectivity by structural features close to the primary binding contacts Jason N. Campbell, Ryan L. Simon, David A Spivak |
92 | Guest-induced chirality in a self-assembled capsule Alessandro Scarso, Julius Rebek, Alexander Shivanyuk, Osamu Hayashida |
93 | Triply-threaded rotaxanes leading to molecular lifts Jovica D. Badjic, J Fraser Stoddart |
94 | Construction of a nanoscale molecular muscle based on molecular recognition Ja-Young Han, J Fraser Stoddart |
95 | Interlocked molecules beyond catenanes and rotaxanes: Investigating supramolecular assistance to covalent synthesis Avril R. Williams, David J. Williams, Andrew J.P. White, J. Fraser Stoddart |
96 | Investigating the potential of tris(2-pyridyl)methane derivatives as carbonic anhydrase mimics Jiachang Gong, Bruce C. Gibb |
97 | Synthesis and self-assembly of benzyl alcohols and benzyl alcohol deep-cavity cavitands Jodie O. Green, Corinne L.D. Gibb, Bruce C. Gibb |
98 | Synthesis and binding studies of three molecular baskets Zachary R. Laughrey, Corinne L.D. Gibb, Tangi Senechal, Bruce C. Gibb |
99 | Magic ring rotaxanes via olefin metathesis Robert H. Grubbs, Stuart J. Cantrill, Andreas F. M. Kilbinger, Andrew W. Waltman, Erin N. Guidry |
100 | Dimeric molecular capsule under redox control Kwangyul Moon, Kaifer Angel |
101 | Enzymological studies of carbon-bound fluorine in intermolecular interactions Khanh C. Hoang, Oana Martin, Sandro Mecozzi |
102 | Formation of a complex dimer assisted by water Feihe Huang, Lev N. Zakharov, Arnold. L. Rheingold, Harry W. Gibson, Jason W. Jones |
103 | Attachment of pyrene fluorophore to silica surfaces via the strongly hydrogen bonding 2-ureido-4-pyrimidone moiety Loretta L. Crowe, Kyril M Solntsev, Laren Tolbert |
104 | Conjugation of poor inhibitors of carbonic anhydrase with surface binding groups: A strategy to improve inhibitor efficiency Bidhan C. Roy, Ryan Hegge, Theresa A. Rosendahl, Xiao Jia, Sanku Mallik |
105 | Preparation of biphenyltetrazole-hydantoins and thiohydantoins as growth hormone secretagogues analogs Rune Severinsen, Jesper Lau, Mikael Begtrup, Michael Ankersen |
106 | Design of triplex-forming molecules Jiansen Li, Yun-Hua Fan, Luis A. Marky, Barry Gold |
107 | Diastereomeric discrimination: Resolution and development of a nonaromatic chiral acid resolving agent with arylamine efficacy J. Luke Gatlin, Edward J. Valente |
108 | A novel type of fluorescent boronic acid that shows large fluorescence intensity changes upon binding with a diol in aqueous solution at physiological pH Binghe Wang, Wenqian Yang, Jun Yan, Greg Springsteen, Susan Deeter |
109 | Calix-peptides: Modular strategy toward polyfunctional receptors and nanoscale assembles Dmitry M. Rudkevich, Heng Xu |
110 | A facile procedure for determining the pKa of weakly acidic pharmaceutical drugs and supramolecular ligands Arno Kraft |
111 | Dimethyl disulfide addition to 1,4-enynes: A new route to 2,5-dialkylthiophenes Lizhi Zhu, Gordon V. Givan, Rachel A. Taylor, Robert E. Minto |
112 | Isolation of a novel pacifigorgiane sesquiterpene Larry G. French, Anthony J. Tracey, Carlos R. Ramirez-Sosa |
113 | Synthesis of carbohydrate derivatives using clean chemistry Rachel N. MacCoss, Paul E. Brennan, Steven V. Ley |
114 | Total synthesis and antileukemic activity of the novel fatty acid 2-methoxy-14-methylpentadecanoic acid Néstor M. Carballeira, Heidyleen Cruz, Elsie A. Orellano, Fernando A. González |
115 | Briarellins J-P and polyanthellin A: New eunicellin-based diterpenes from the Caribbean gorgonian coral Briareum polyanthes Claudia A. Ospina, Abimael D. Rodríguez |
116 | Synthesis and bioactivity of erebusinone, a pigment from the antarctic sponge Isodictya erinacea Young Chul Park, Bill J. Baker |
117 | Design, synthesis, and evaluation of an enediyne with a new activation mechanism Martin F Semmelhack, Lingyun Wu, Robert A. Pascal Jr., Douglas M. Ho |
118 | Nonactin biosynthesis: Nonactin is cleaved by a serine esterase-like protein encoded by the nonactin resistance gene, nonR James E. Cox, Nigel D. Priestley |
119 | Photoreversible serine protease inhibitor synthesis and application Junhai Yang, Ned A. Porter |
120 | Photosensitive serine protease inhibitors based on the naphthalene ring system Birgit Reeves, Ned A. Porter |
121 | Synthesis of a new series of flavonoids Michael E. McKendall, Tasha P. Smith, Maryam Foroozesh |
122 | Chemical synthesis of a carbohydrate-based hydroxamic acid inhibitor of LpxCs Xuechen Li, Taketo Uchiyama, Ole Hindsgaul |
123 | Detection of dsDNA in homogeneous solution by hairpin polyamide-tetramethyl rhodamine conjugates Victor C. Rucker, Alex R. Dunn, Shantanu Sharmu, H. B. Gray, Jay R. Winkler, Peter B. Dervan |
124 | Synthesis of two analogs of 8-oxo-2'-deoxyguanosine, a potent promutagen Michelle Hamm, Courtney Hoey, Waitman Aumann |
125 | Systematic investigations of the effect of pH, urea, and neighboring amino acids on the random coil a-proton chemical shift of alanine in short peptides Sonya L. McKay, Abby M. Maranda, Elizabeth A. Carlisle |
126 | Synthesis and characterizations of some novel Horner-Wadsworth-Emmons reagents Guifa Su, Ling Pan, Longmei Zeng |
127 | Synthesis of an orthogonally protected triester platform related to marine cyclopeptides Laurent Trembleau, Wook-Dong Cho, Byron W. Purse, Julius Rebek Jr. |
128 | Design of novel fluorescence energy transfer cassettes utilizing a nucleobase as part of the donor Guan-Sheng Jiao, Lars H. Thoresen, Kevin Burgess |
129 | Novel synthesis and characterization of b-selenolo[2,3-b]pyrrolyl-L-alanine ([6,7]SeTrp) and its potential use in the elucidation of protein structure and dynamics Duane M. Hatch, Louis A Silks III, Jeffrey O. Boles |
130 | Efficient large-scale synthesis of picolinic acid derived Ni(II)complexes of glycine as new and synthetically efficient equivalents of nucleophilic glycine Vadim A. Soloshonok, Hisanori Ueki, Trevor K. Ellis, Collin H. Martin |
131 | Efficient method for removal of ruthenium by-products from olefin metathesis reactions Jong Hyun Cho, B. Moon Kim |
132 | Synthesis and structure of new acyclic analogs of nucleotides containing a 1,2- or 1,3-alkadienic skeleton Valery K. Brel, Peter J Stang |
133 | Synthesis of purine monomers for a-helical peptide nucleic acids Philip Garner, Michelle M. Adams |
134 | Design of heterocomplexes for supramolecular polymers and surface functionalization Godefridus B.W.L. Ligthart, Rint P. Sijbesma, E.W. Meijer |
135 | A geomorphic classification of antibody binding sites K. N. Houk, Michelle Lee, Julie Schallhorn, Keiki Sugimoto, Andrew G. Leach |
136 | A new strategy to induce g-turn: Peptides composed of alternating a-aminoxy acids and a-amino acids Wei Li, Dan Yang |
137 | Cross-linked hemoglobin dye conjugates for photodynamic therapy Claudia M. Davila, David S. Crumrine, Kenneth Olsen |
138 | b 2,2-Aminoxy acids: A new building block for turns and helices Yu-Hui Zhang, Dan Yang, Nian-Yong Zhu |
139 | Highly specific HPLC-UV method for the determination of cysteine and related aminothiols in biological samples Venkataraman Amarnath, Kapil Amarnath, Holly L. Valentine, William M. Valentine, Kalyani Amarnath |
140 | Quinomethionate acting as a photoinducible DNA cleaving agent Jian Ying Qi, Albert S. C. Chan, Tianhu Li |
141 | Synthesis and conductance study of trans-1,2-cyclopentane dicarboxamide linked gramicidin A dimers David S. Crumrine, Shasikala Narayan, Courtney Williams, Samuel Cukierman |
142 | Synthesis and application of polymer-supported (-)-sparteine as an external chiral ligand Madugula S. R. Murty, John M. Rimoldi |
143 | Synthesis of polymer-bound silyl azide for solid-phase organic synthesis Richard T. Taylor, Matthew W. Bedore, Jennifer A. Fisher |
144 | Tandem Petasis-Ugi multicomponent condensation reactions: A practical preparation of multidimensional libraries Laura West, David E. Portlock, Ryszard Ostaszewski, Dinabandhu Naskar |
145 | Reactivity and synthesis of substituted furanones and a novel approach to optically active derivatives applied in quorum-sensing inhibition bioassays Tobias Persson, John Nielsen, Thomas Hjelmgaard |
146 | Sonogashira chemistry for solid-phase organic synthesis Judit Tulla-Puche, George Barany |
147 | Suzuki cross-coupling using glass beads technology Kokovi M. Lawson Daku, Jonathan M.J. Williams, Roger F. Newton |
148 | Peptides as precursors to peptidomimetics: Novel approach to class B streptogramin antibiotics Jennifer L. Robinson, Shelli R. McAlpine, Enrique V. Azevedo |
149 | Catalytic asymmetric cylcopropanation using polymer-supported rhodium(II) catalysts Sambasiva R. Poreddy, John M. Rimoldi |
150 | High-throughput synthesis of anilide libraries on solid support Moustafa E. El-Araby, Helen Guo, Richard S. Pottorf, Mark R. Player |
151 | Novel antibiotics: Macrocyclic peptides designed to trap the Holliday junction Lisa A. Liotta, Jason Smith, Shelli R. McAlpine |
152 | A novel solid-phase synthesis of cyclic sulfonamide analogs of 4-hydroxyquinolinones Caiding Xu, Ashok Bhandari, Christopher P. Holmes |
153 | A solid-phase synthesis of diacylglycerol-lactones in macrokans as a prelude to the synthesis of protein kinase C isozyme-specific ligands by a combinatorial approach Dehui Duan, Victor E. Marquez |
154 | A facile parallel synthesis of indazoles with three-point diversities on solid support Y. Sarah Dong, Jillian Basinger, Ashok Bhandari, Christopher P. Holmes |
155 | A general solid-phase synthesis of 4-substituted quinolinones via a Pd-catalyzed negishi cross-coupling reaction Caiding Xu, Lydie Yang, Ashok Bhandari, Christopher P. Holmes |
156 | A novel method for mono-N-alkylation of primary amines and its application to synthesis of small organic compound libraries on the ACT solution-phase synthesizer, “The Solution” Eugene Campian, HupChew Wong, Mahendra Menakuru, Justin Rogosky, Leslie Craddock, Jim Shannon, Hossain Saneii, Boliang Lou |
157 | Combinatorial strategies for the synthesis of vancomycin derivatives with improved antibacterial properties Aveline Yim, Martin Wills |
158 | Solid-phase synthesis of a library of hydroxyproline derivatives Anne L. Vergnon, Richard S. Pottorf, Mark R. Player |
159 | Polymer-bound oxoammonium salt of TEMPO: A novel reagent for selective oxidation of alcohols Sukanta Bhattacharyya, Lanchi Vo, Tejal Parekh, Jeff Labadie |
160 | Utilization of 400–500-micron polystyrene beads for the preparation of encoded combinatorial libraries Thuy X. H. Le, Huarong Ma, Tao Guo, Vinh Tran, Doug Hobbs, Peter Kieselback, Ed Heebner |
161 | ACTU: A novel coupling agent for polymer-bound HOBt active esters Tejal Parekh, Sukanta Bhattacharyya, Owen Gooding, Thomas J Lindberg, Jeff W. Labadie |
162 | Removal of amines from solution: A comparison of solid-supported scavengers A. J. Mendonca, Andrew F Coffey, John W Davies, Peter A Marsh, M. I. Richards, B. Thomas, D. J. Woodward, F.P. Warner |
163 | High-throughput microwave-accelerated combinatorial synthesis: A plate-based approach John J Lord, Christopher R. Sarko |
164 | Solid-phase synthesis of di- and trisubstituted N-acyl ureas: A novel approach Jacob Ravn, Jesper Lau, Mikael Begtrup, Michael Ankersen |
165 | Highly regioselective parallel solid-phase synthesis of new tetracyclic 1,3,5-triazino[1,2-a]benzimidazoles Cornelia E. Hoesl, Adel Nefzi, Richard A. Houghten |
166 | Lead-generation libraries based on a 1,2,5-thiadiazole-1-oxide template Richard D. Gless Jr., Maureen M. McKenna, Michael T. Keller, Stephen C. Smith, Christopher Mathews |
167 | Lead-generation libraries based on a 3-amino-1,4-oxo-1,2,5-thiadiazole acetamide template Richard D. Gless Jr., Maureen M. McKenna, Michael T. Keller, Stephen C. Smith |
168 | New technique to parallel solution-phase synthesis of esters by solid-supported sulfonyl chloride cartridge Shahnaz Ghassemi, Peter Rahn, Michael Webb |
169 | Synthesis of an isoxazolinopyrrole library Sung Hee Hwang, Mark J. Kurth |
Symposium Grid -- Division of Organic Chemistry -- Session Listing
The 225th ACS National Meeting, New Orleans, LA, March 23-27, 2003